Novo-bromazepam: Full Drug Profile
Novo-bromazepam - General Information
One of the benzodiazepines that is used in the treatment of anxiety disorders. [PubChem] It is a Schedule IV drug in the U.S. and Canada and under the Convention on Psychotropic Substances.
Pharmacology of Novo-bromazepam
Novo-bromazepam is a lipophilic, long-acting benzodiazepine and with sedative, hypnotic, anxiolytic and skeletal muscle relaxant properties. It does not possess any antidepressant qualities. Novo-bromazepam shares with other benzodiazepines the risk of abuse, misuse, psychological and/or physical dependence. According to many psychiatric experts Novo-bromazepam has a greater abuse potential than other benzodiazepines because of fast resorption and rapid onset of action.
Additional information about Novo-bromazepam
- Novo-bromazepam Indication
For the short-term treatment of insomnia, short-term treatment of anxiety or panic attacks, if a benzodiazepine is required, and the alleviation of the symptoms of alcohol- and opiate-withdrawal.
- Mechanism Of Action
- Novo-bromazepam binds to the GABA receptor GABAA, causing a conformational change and increasing inhibitory effects of GABA. Other neurotransmitters are not influenced.
- Generic Name
- Bromazepam
- Synonyms
- 7-Bromo-5-(2-pyridyl)-3H-1,4-benzodiaxepin-2(1H)-one; 7-Bromo-5-(2-pyridyl)-3H-1,4-benzodiazepin-2(1H)-one; Bromazepamum [inn-latin]
- Drug Category
- Benzodiazepines; Hypnotics and Sedatives
- Drug Type
- Small Molecule; Illicit; Approved
- Other Brand Names containing Bromazepam
- Apo-Bromazepam; Calmepam; Compedium; Compendium; Creosedin; Durazanil; Gen-Bromazepam; Lectopam; Lekotam; Lexaurin; Lexilium; Lexomil; Lexotan; Lexotanil; Normoc; Novo-bromazepam; Nu-Bromazepam; Ultramidol; Somalium;
- Absorption
- Bioavailability is 84% following oral administration.
- Biotransformation
- Hepatically, via oxidative pathways (via an enzyme belonging to the Cytochrome P450 family of enzymes).
- Half Life
- 10-20 hours
- Dosage Forms of Novo-bromazepam
- Tablet Oral
- Chemical IUPAC Name
- 7-bromo-5-pyridin-2-yl-1,3-dihydro-1,4-benzodiazepin-2-one
- Chemical Formula
- C14H10BrN3O
- Bromazepam on Wikipedia
- https://en.wikipedia.org/wiki/Bromazepam
- Organisms Affected
- Humans and other mammals
