Colum: Full Drug Profile
Colum - General Information
Colum is a post-ganglionic parasympathetic inhibitor. It decreases gastric acid and pepsin secretion and suppresses spontaneous contractions of the colon. Colum diminishes gastric acid and pepsin secretion. Colum also suppresses spontaneous contractions of the colon. Pharmacologically, it is a post-ganglionic parasympathetic inhibitor. It has not been shown to be effective in contributing to the healing of peptic ulcer, decreasing the rate of recurrence, or preventing complications.
Pharmacology of Colum
Colum diminishes gastric acid and pepsin secretion. Colum also suppresses spontaneous contractions of the colon. Pharmacologically, it is a post-ganglionic parasympathetic inhibitor.
Additional information about Colum
- Colum Indication
For use as adjunctive therapy in the treatment of peptic ulcer. It has not been
- Mechanism Of Action
- Colum is a post-ganglionic parasympathetic inhibitor. It decreases gastric acid and pepsin secretion and suppresses spontaneous contractions of the colon.
- Generic Name
- Mepenzolate
- Synonyms
- 1-Methyl-3-piperidyl benzilate methyl bromide; Mepenzolate bromide; Mepenzolic acid; N-Methyl-3-piperidyl benzilate methyl bromide; N-Methyl-3-piperidyldiphenylglycolate methobromide
- Drug Category
- Anticholinergic Agents; Parasympatholytics
- Drug Type
- Small Molecule; Approved
- Other Brand Names containing Mepenzolate
- Cantil; Cantilaque; Cantilon; Cantril; Colibantil; Colopiril; Colum; Delevil; Eftoron; Gastropidil; Mepenzolon; Tralanta; Trancolon;
- Absorption
- Between 3 and 22% of an orally administered dose is excreted in the urine over a 5-day period, with the majority of the radioactivity appearing on Day 1. The remainder appears in the next 5 days in the feces and presumably has not been absorbed.
- Toxicity (Overdose)
- The signs and symptoms of overdosage are headache; nausea; vomiting; blurred vision; dilated pupils; hot, dry skin; dizziness; dryness of the mouth; difficulty in swallowing; and CNS stimulation. A curare-like action may occur (i.e., neuromuscular blockade leading to muscular weakness and possible
- Dosage Forms of Colum
- Tablet Oral
- Chemical IUPAC Name
- (1,1-dimethylpiperidin-1-ium-3-yl) 2-hydroxy-2,2-di(phenyl)acetate
- Chemical Formula
- C21H26NO3
- Organisms Affected
- Humans and other mammals
