Patanol: Full Drug Profile
Patanol - General Information
Used to treat allergic conjunctivitis (itching eyes), olopatadine inhibits the release of histamine from mast cells. It is a relatively selective histamine H1 antagonist that inhibits the in vivo and in vitro type 1 immediate hypersensitivity reaction including inhibition of histamine induced effects on human conjunctival epithelial cells.
Pharmacology of Patanol
Used to treat allergic conjunctivitis (itching eyes), olopatadine inhibits the release of histamine from mast cells. It is a relatively selective histamine H1 antagonist that inhibits the in vivo and in vitro type 1 immediate hypersensitivity reaction including inhibition of histamine induced effects on human conjunctival epithelial cells.
Patanol for patients
Patanol Interactions
No information provided.
Patanol Contraindications
PATANOL (olopatadine hydrochloride ophthalmic solution) 0.1% is contraindicated in persons with a known hypersensitivity to olopatadine hydrochloride or any components of PATANOL.
Additional information about Patanol
- Patanol Indication
For the treatment of the signs and symptoms of allergic conjunctivitis.
- Mechanism Of Action
- Patanol is a selective histamine H1 antagonist and binds to the histamine H1 receptor. This blocks the action of endogenous histamine, which subsequently leads to temporary relief of the negative symptoms brought on by histamine. Patanol is devoid of effects on alpha-adrenergic, dopamine and muscarinic type 1 and 2 receptors.
- Generic Name
- Olopatadine
- Drug Category
- Anti-Allergic Agents; Anti-Inflammatory Agents, Non-Steroidal; Antihistamines; Histamine H1 Antagonists
- Drug Type
- Small Molecule; Approved
- Other Brand Names containing Olopatadine
- Olopatadine Hydrochloride; Patanol;
- Absorption
- Ophthalmic use of olopatadine usually does not produce measurable plasma concentrations.
- Biotransformation
- The mono-desmethyl and the N-oxide metabolites have been detected at low concentrations in the urine.
- Half Life
- 3 hours
- Dosage Forms of Patanol
- Liquid Ophthalmic
- Chemical IUPAC Name
- 2-[(11Z)-11-(3-dimethylaminopropylidene)-6H-benzo[c][2]benzoxepin-2-yl]acetic acid
- Chemical Formula
- C21H23NO3
- Olopatadine on Wikipedia
- https://en.wikipedia.org/wiki/Olopatadine
- Organisms Affected
- Humans and other mammals
