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Definition of Antiandrogen

Medically reviewed by Min Clinic Staff | Updated: January 2026

Antiandrogen: A drug that blocks the action of androgens (male sex hormones). Antiandrogens are sometimes used in the treatment of prostate cancer. The antiandrogens currently available include flutamide (Eulexin), bicalutamide (Casodex), and nilutamide (Nilandron).